Entry ID |
Original Release date |
Data summary |
Entry Title |
Citation Title |
Authors |
51480 |
2023-11-17 |
Chemical Shifts: 1 set |
Androgen Receptor NTD |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
51479 |
2022-09-30 |
Chemical Shifts: 1 set |
Androgen Receptor AF1star |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
51476 |
2023-11-17 |
Chemical Shifts: 1 set |
Androgen Receptor C-terminal NTD |
Rational optimization of a transcription factor activation domain inhibitor
|
Albert Escobedo, Alessandro Ruffoni, Antoni Riera, Borja Mateos, C Adriana A Banuelos, Carla Garcia-Cabau, Carolina Sanchez-Zarzalejo, Cristina Batlle, David Meierhofer, Denes Hnisz, Elzbieta Szulc, Hannes Dockx, Harpreet Kaur, Isabelle Brun-Heath, Jesus Garcia, Jiaqi Zhu, Jon K Obst, Jordann Smak, Jun Wang, Karina Pombo-Garcia, Levente Zodi, Lidia Bardia, Marianne D Sadar, Marta Frigole-Vivas, Mateusz Biesaga, Michael Lewis, Mireia Pesarrodona, Nasrin R Mawji, Paula Martinez-Cristobal, Paul Robustelli, Salvador Ventura, Shaon Basu, Stase Bielskute, Teresa Tam, Travis H Stracker, Xavier Salvatella, Xavier Verdaguer |
34491 |
2021-01-26 |
Chemical Shifts: 1 set |
Cortistatin analog with improved immunoregulatory activity |
Structure-based design of a Cortistatin analogue with immunomodulatory activity in models of inflammatory bowel disease
|
A Escola, A Riera, A Rol, B Ponsati, E Aragon, E Gonzalez-Rey, E Puig, J Farrera-Sinfreu, J Fernandez-Carneado, M Delgado, M J Macias, M Valles-Miret, P Martin-Malpartida, T Todorovski, X Verdaguer |
27548 |
2018-11-15 |
Chemical Shifts: 1 set |
Ressonance assignments for the human Smad5 MH1 domain |
TGIF1 homeodomain interacts with Smad MH1 domain and represses TGF-beta signaling.
|
Agnieszka Konkol, Antoni Riera, Carles Torner, David Sunol, Eric Aragon, Ewelina Guca, Jorge Cordero, Lidia Ruiz, Maria J Macias, Pau Martin-Malpartida |
27461 |
2018-07-17 |
Chemical Shifts: 1 set |
Human TGIF1 c-term domain |
TGIF1 homeodomain interacts with Smad MH1 domain and represses TGF-beta signaling.
|
Agnieszka Konkol, Antoni Riera, Carles Torner, David Sunol, Eric Aragon, Ewelina Guca, Jorge Cordero, Lidia Ruiz, Maria J Macias, Pau Martin-Malpartida |
26794 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp6,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
26799 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp6,L-Msa7,D-Trp8, L-Dfp11-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
26798 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp11,L-Msa7,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
26797 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp6,L-Msa7,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
26796 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp11,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |
26795 |
2016-08-31 |
Chemical Shifts: 1 set |
NMR Assignment of L-Dfp7,D-Trp8-SRIF |
Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3',5'difluorophenyl)-alanine
|
Alvaro Rol, Antoni Riera, Berta Ponsati, Eric Aragon, Jimena Fernandez-Carneado, Maria J Macias, Mariona Valles-Miret, Pablo Martin-Gago, Pau Martin-Malpartida, Toni Todorovski, Xavier Verdaguer |