Entry ID |
Original Release date |
Data summary |
Entry Title |
Citation Title |
Authors |
51472 |
2022-10-19 |
Chemical Shifts: 1 set |
Backbone amide chemical shifts for PBRM1-BD2 |
Selective and Cell-Active PBRM1 Bromodomain Inhibitors Discovered through NMR Fragment Screening
|
Brayden P Strohmier, Brian C Smith, Brian F Volkman, Christopher J Goetz, Davin R Jensen, Emily C Dykhuizen, Francis C Peterson, Karina L Bursch, Mallory K Roach, Maya E Blau, Michael D Olp, Raymundo Nunez, Sandra C Ordonez-Rubiano, Shifali Shishodia, Tyler G Fenske |
51450 |
2022-10-19 |
Chemical Shifts: 1 set |
Backbone amide chemical shifts for PBRM1-BD2 bound to 5-Chloro-2-(3-methylphenyl)-2,3-dihydroquinazolin-4(1H)-one |
Selective and Cell-Active PBRM1 Bromodomain Inhibitors Discovered through NMR Fragment Screening
|
Brayden P Strohmier, Brian C Smith, Brian F Volkman, Christopher J Goetz, Davin R Jensen, Emily C Dykhuizen, Francis C Peterson, Karina L Bursch, Mallory K Roach, Maya E Blau, Michael D Olp, Raymundo Nunez, Sandra C Ordonez-Rubiano, Shifali Shishodia, Tyler G Fenske |
27706 |
2018-12-19 |
Chemical Shifts: 1 set |
EZH2 SANT1 |
The EZH2 SANT1 domains is a histone reader domain providing sensitivity to the modification state of the H4 tail
|
Catherine A Musselman, Chris Coble, Emily C Dykhuizen, Jiachen Liu, Katayoun Varzavand, Katelyn E Connelly, Tyler M Weaver |
27616 |
2018-12-17 |
Chemical Shifts: 1 set |
Backbone 1H, 13C, and 15N Chemical Shift Assignments for CBX8 chromodomain |
Engagement of DNA and H3K27me3 by the CBX8 chromodomain drives chromatin association.
|
Aktan Alpsoy, Brian X Gu, Catherine A Musselman, Emily C Dykhuizen, Katelyn E Connelly, Tyler M Weaver |